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bioRxiv · 10.1101/2020.08.14.251207

SRSF protein kinases 1 and 2 are essential host factors for human coronaviruses including SARS-CoV-2

Abstract

While vaccines are vital for preventing COVID-19 infections, it is critical to develop new therapies to treat patients who become infected. Pharmacological targeting of a host factor required for viral replication can suppress viral spread with a low probability of viral mutation leading to resistance. In particular, host kinases are highly druggable targets and a number of conserved coronavirus proteins, notably the nucleoprotein (N), require phosphorylation for full functionality. In order to understand how targeting kinases could be used to compromise viral replication, we used a combination of phosphoproteomics and bioinformatics as well as genetic and pharmacological kinase inhibition to define the enzymes important for SARS-CoV-2 N protein phosphorylation and viral replication. From these data, we propose a model whereby SRPK1/2 initiates phosphorylation of the N protein, which primes for further phosphorylation by GSK-3/{beta} and CK1 to achieve extensive phosphorylation of the N protein SR-rich domain. Importantly, we were able to leverage our data to identify an FDA-approved kinase inhibitor, Alectinib, that suppresses N phosphorylation by SRPK1/2 and limits SARS-CoV-2 replication. Together, these data suggest that repurposing or developing novel host-kinase directed therapies may be an efficacious strategy to prevent or treat COVID-19 and other coronavirus-mediated diseases.

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BibTeXRIS

Heaton, B. E., Trimarco, J. D., Hamele, C. E., Harding, A. T., Tata, A., Zhu, X., Tata, P. R., Smith, C. M., Heaton, N. S.. 2020-08-14. SRSF protein kinases 1 and 2 are essential host factors for human coronaviruses including SARS-CoV-2. https://doi.org/10.1101/2020.08.14.251207

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