@misc{indiciae6f3a98a59fd7, title = {Open-science discovery of DNDI-6510, a compound that addresses genotoxic and metabolic liabilities of the COVID Moonshot SARS-CoV-2 Mpro lead inhibitor}, author = {Griffen, E. J. and Fearon, D. and McGovern, B. L. and Koekemoer, L. and Balcomb, B. H. and Szommer, T. and Fate, G. and Robinson, R. P. and Lefker, B. A. and Duberstein, S. and Lahav, N. and Braillard, S. and Vangeel, L. and Laporte, M. and Charvillon, F. B. and MacLeod, A. K. and Wells, A. and Garner, P. and Knight, R. and Rees, P. and Simon, A. and Jochmans, D. and Neyts, J. and Read, K. D. and Barr, H. and Robinson, M. and Lee, A. A. and London, N. and Chodera, J. and von Delft, F. and White, K. M. and Perry, B. and Sjo, P. and von Delft, A. R.}, year = {2025}, doi = {10.1101/2025.06.16.660018}, url = {https://www.biorxiv.org/content/10.1101/2025.06.16.660018v1}, note = {Source identifier: 10.1101/2025.06.16.660018} }