TY  - RPRT
TI  - Discovery and characterization of FX-909, a covalent inverse agonist of PPARG rationally designed to impose a powerful repressive bias in PPARG for the treatment of PPARG/RXRA-activated muscle-invasive urothelial cancers
AU  - Stuckey, J. I.
AU  - Mertz, J. A.
AU  - Wilson, J. E.
AU  - Williamson, K. E.
AU  - Li, Y.
AU  - Kuljanin, M.
AU  - DeLaBarre, B.
AU  - Chenail, G.
AU  - Nguyen, P. A.
AU  - Bailey, C. M.
AU  - Motley, W. M.
AU  - Audia, J. E.
AU  - Sims, R. J.
PY  - 2025
DO  - 10.1101/2025.05.08.652848
UR  - https://www.biorxiv.org/content/10.1101/2025.05.08.652848v1
ID  - 10.1101/2025.05.08.652848
ER  -