@misc{indiciae8c24d9f9f821, title = {Shifting the PPARγ conformational ensemble towards a transcriptionally repressive state improves covalent inhibitor efficacy}, author = {Arifova, L. and MacTavish, B. S. and Laughlin, Z. and Karadi Girdhar, M. N. and Shang, J. and Li, M.-H. and Yu, X. and Zhu, D. and Kamenecka, T. M. and Kojetin, D.}, year = {2025}, doi = {10.1101/2025.03.04.640448}, url = {https://www.biorxiv.org/content/10.1101/2025.03.04.640448v1}, note = {Source identifier: 10.1101/2025.03.04.640448} }